SCHEMBL206098

SCHEMBL206098

CN(C)C1(c2cccs2)CCC(NC(=O)CCCC(=O)N2CC=C(c3ccc(F)cc3)CC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.41
MAPT P10636 3/20 0.39
ALDH1A1 P00352 3/20 0.39
ALOX15 P16050 2/20 0.39
NPC1 O15118 1/20 0.39
HPGD P15428 1/20 0.39
CASP3 P42574 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
PARP1 P09874 4/20 0.39
PARP2 Q9UGN5 1/20 0.39
NAMPT P43490 5/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ENPP2 Q13822 1/20 0.37
KDM4E B2RXH2 3/20 0.36
OPRM1 P35372 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL207139 0.87 OPRM1 (0.37) MAPK1MAPTALDH1A1ALOX15NPC1
SCHEMBL206892 0.81 ALDH1A1 (0.48) MAPTALDH1A1NPC1HPGDRAB9A
SCHEMBL4074077 0.80 OPRM1 (0.51) NPC1RAB9ASMN1; SMN2OPRM1OPRL1
SCHEMBL5477680 0.78 OPRM1 (0.41) MAPK1MAPTALDH1A1ALOX15NPC1
SCHEMBL4074080 0.78 OPRM1 (0.51) NPC1RAB9AOPRM1OPRL1
SCHEMBL4079677 0.77 OPRM1 (0.47) NPC1RAB9AOPRM1OPRL1
SCHEMBL206590 0.76 MEN1 (0.47) MAPTALDH1A1ALOX15NPC1HPGD
SCHEMBL4046091 0.75 ACKR3 (0.50) ALDH1A1MEN1KMT2AOPRM1OPRL1
SCHEMBL205169 0.74 SIGMAR1 (0.41) MAPK1MAPTALDH1A1ALOX15NPC1
SCHEMBL4079674 0.74 OPRM1 (0.45) NPC1RAB9AOPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088763-B2 e.g. N-[1-(2,6-dichloro-benzyl)-pyrrolidin-3-yl]-N'-[4-dimethylamino-4-(4-methyl-benzyl)-cyclohexyl]-succinamide; noradrenaline and serotonin reuptake ihibitor; opioid ORL-1 receptor ligand; analgesic, antidepressant, anxiolytic agent, neurodegenerative diseases GRUENENTHAL GMBH (DE) 2012-01-03 US claimed
US-8088763-B2 e.g. N-[1-(2,6-dichloro-benzyl)-pyrrolidin-3-yl]-N'-[4-dimethylamino-4-(4-methyl-benzyl)-cyclohexyl]-succinamide; noradrenaline and serotonin reuptake ihibitor; opioid ORL-1 receptor ligand; analgesic, antidepressant, anxiolytic agent, neurodegenerative diseases GRUENENTHAL GMBH (DE) 2012-01-03 US disclosed