SCHEMBL20627367

SCHEMBL20627367

CC(C)Cc1cccc2c1CCC(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.43
OPRK1 P41145 2/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
NPC1 O15118 1/20 0.42
MAPK13 O15264 1/20 0.42
MAPK12 P53778 1/20 0.42
MAPK11 Q15759 1/20 0.42
MAPK14 Q16539 1/20 0.42
KCNH2 Q12809 2/20 0.42
DRD2 P14416 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
CHRM2 P08172 1/20 0.42
CYP3A4 P08684 1/20 0.42
ADRA2A P08913 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
ADRA2B P18089 1/20 0.42
DRD1 P21728 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20627220 0.86 DRD2 (0.56) HTR1AOPRK1KCNH2DRD2KDM4E
SCHEMBL9911041 0.83 HTR1A (0.49) HTR1AOPRK1ADRB2ADRB1NPC1
SCHEMBL17969095 0.80 NPC1 (0.47) HTR1AOPRK1ADRB2ADRB1NPC1
SCHEMBL19386411 0.78 HTR1A (0.45) HTR1AOPRK1ADRB2ADRB1NPC1
SCHEMBL427050 0.76 NPC1 (0.43) HTR1AOPRK1ADRB2ADRB1NPC1
SCHEMBL12285526 0.76 GABRA1 (0.44) HTR2AHTR2BGABRA1GABRB2
SCHEMBL12546146 0.76 NPC1 (0.46) HTR1AOPRK1ADRB2ADRB1NPC1
SCHEMBL426989 0.75 NPC1 (0.42) HTR1AOPRK1ADRB2ADRB1NPC1
SCHEMBL12020822 0.74 DRD2 (0.46) HTR1AOPRK1ADRB2ADRB1NPC1
SCHEMBL19772860 0.73 GABRA1 (0.42) HTR1ADRD2HTR2AHTR2BGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3224252-B1 SUBSTITUTED OXAZOLE- AND THIAZOLE-BASED CARBOXAMIDE AND UREA DERIVATIVES AS VANILLOID RECEPTOR LIGANDS II MEDIFRON DBT INC (KR) 2019-01-09 EP disclosed