SCHEMBL2062932

SCHEMBL2062932

CCOC(=O)Cc1c(Cl)ncnc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 4/20 0.43
LMNA P02545 1/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
MAPK1 P28482 2/20 0.42
TDP1 Q9NUW8 3/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
RAB9A P51151 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
MAPT P10636 2/20 0.40
USP2 O75604 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GAA P10253 2/20 0.39
MGAM O43451 1/20 0.39
SI P14410 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8692811 0.92 KDM4E (0.43) SMN1; SMN2KDM4ELMNAKMT2AMEN1
SCHEMBL12590746 0.89 SMN1; SMN2 (0.46) SMN1; SMN2KDM4ELMNAKMT2AMEN1
SCHEMBL2062770 0.81 ALDH1A1 (0.42) SMN1; SMN2KDM4ELMNAKMT2AMEN1
SCHEMBL12590776 0.81 CYP1A2 (0.44) SMN1; SMN2TDP1L3MBTL1TSHRHSD17B10
SCHEMBL5844147 0.80 MAPK1 (0.46) KDM4ELMNAKMT2AMEN1MAPK1
SCHEMBL1748473 0.80 MAPK1 (0.46) KDM4ELMNAKMT2AMEN1MAPK1
SCHEMBL2063964 0.80 MAPK1 (0.46) SMN1; SMN2KDM4ELMNAKMT2AMEN1
SCHEMBL30959611 0.79 SMN1; SMN2 (0.39) SMN1; SMN2LMNAKMT2AMEN1MAPK1
SCHEMBL1055154 0.79 MAPK1 (0.53) SMN1; SMN2KDM4ELMNAKMT2AMEN1
SCHEMBL12000330 0.78 KDM4E (0.41) SMN1; SMN2KDM4ELMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118440011-A Purification method of 4, 6-dichloropyrimidine or derivative thereof 诚达药业股份有限公司 2024-08-06 CN disclosed
CN-118440010-A Preparation method of 4, 6-dichloro-5-pyrimidine acetaldehyde 诚达药业股份有限公司 2024-08-06 CN disclosed
CN-102216302-B Akt and p70 s6 kinase inhibitors LILLY CO ELI 2013-08-21 CN disclosed
EP-2358710-B1 AKT AND P70 S6 KINASE INHIBITORS LILLY CO ELI (US) 2012-08-15 EP disclosed
US-8148387-B2 AKT and P70 S6 kinase inhibitors ELI LILLY AND COMPANY (US) 2012-04-03 US disclosed
US-8148387-B2 AKT and P70 S6 kinase inhibitors ELI LILLY AND COMPANY (US) 2012-04-03 US disclosed
US-8148387-B2 AKT and P70 S6 kinase inhibitors ELI LILLY AND COMPANY (US) 2012-04-03 US disclosed
CN-102216302-A Akt and p70 s6 kinase inhibitors LILLY CO ELI 2011-10-12 CN disclosed
US-7968536-B2 Heterocyclic compounds useful as RAF kinase inhibitors MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-06-28 US disclosed
US-7968536-B2 Heterocyclic compounds useful as RAF kinase inhibitors MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-06-28 US disclosed
WO-2010056563-A1 AKT AND P70 S6 KINASE INHIBITORS ELI LILLY AND COMPANY (US) 2010-05-20 WO disclosed
US-20100120801-A1 AKT AND P70 S6 KINASE INHIBITORS ELI LILLY AND COMPANY 2010-05-13 US disclosed
US-20100120801-A1 AKT AND P70 S6 KINASE INHIBITORS ELI LILLY AND COMPANY 2010-05-13 US disclosed
US-20100120801-A1 AKT AND P70 S6 KINASE INHIBITORS ELI LILLY AND COMPANY 2010-05-13 US disclosed
US-20090005359-A1 Heterocyclic Compounds Useful as RAF Kinase Inhibitors SUNESIS PHARMACEUTICALS, INC (US) 2009-01-01 US disclosed
US-20090005359-A1 Heterocyclic Compounds Useful as RAF Kinase Inhibitors SUNESIS PHARMACEUTICALS, INC (US) 2009-01-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100120801-A1 AKT AND P70 S6 KINASE INHIBITORS RPS6KA6, RPS6KA1, MTOR SMN1; SMN2 3551/4885KDM4E 2390/4885LMNA 4229/4885
US-20090005359-A1 Heterocyclic Compounds Useful as RAF Kinase Inhibitors BRAF, RAF1, ARAF SMN1; SMN2 4436/4885KDM4E 2207/4885LMNA 3257/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.