SCHEMBL20632129

SCHEMBL20632129

Cc1ccncc1-c1ccc(N)c(C)n1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 4/20 0.43
CYP11B1 P15538 5/20 0.42
CYP11B2 P19099 5/20 0.42
CYP1A2 P05177 2/20 0.39
CYP2E1 P05181 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C8 P10632 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2A6 P11509 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2B6 P20813 2/20 0.39
CYP2C19 P33261 2/20 0.39
PDE10A Q9Y233 1/20 0.38
PDE2A O00408 1/20 0.38
MAP4K1 Q92918 5/20 0.38
CLK2 P49760 2/20 0.38
DYRK1A Q13627 2/20 0.38
CLK3 P49761 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11909828 0.79 MAP2K3 (0.46) ABL1MAP4K1
SCHEMBL16835968 0.74 CYP1A2 (0.46) ABL1CYP11B1CYP11B2CYP1A2CYP2E1
SCHEMBL22808268 0.73 CDK2 (0.58) ABL1CYP11B1CYP11B2CYP1A2CYP2E1
SCHEMBL16835877 0.72 CYP2A6 (0.57) ABL1CYP1A2CYP3A4CYP2A6CYP2C19
SCHEMBL11241124 0.72 ROCK2 (0.43) ABL1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL29988790 0.72 TDO2 (0.49) ABL1CYP11B1CYP11B2CYP1A2CYP2E1
SCHEMBL3421743 0.72 TDO2 (0.49) ABL1CYP11B1CYP11B2CYP1A2CYP2E1
SCHEMBL30309922 0.72 LCK (0.46) ABL1CYP11B1CYP11B2CYP1A2CYP2E1
SCHEMBL15784053 0.72 LCK (0.46) ABL1CYP11B1CYP11B2CYP1A2CYP2E1
SCHEMBL24667225 0.71 CYP2A6 (0.56) CYP11B1CYP11B2CYP1A2CYP2A6PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2997029-B1 SUBSTITUTED BRIDGED UREA ANALOGS AS SIRTUIN MODULATORS GLAXOSMITHKLINE LLC (US) 2019-01-09 EP disclosed