SCHEMBL20640975

SCHEMBL20640975

C=CC[C@H](O)c1c(F)cccc1F

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.33
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
HRH3 Q9Y5N1 1/20 0.31
ERN1 O75460 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20645990 1.00 CES2 (0.40) CES2CES1CYP2C19SMN1; SMN2HPGD
SCHEMBL20646071 0.82 CYP2C19 (0.31) CYP2C19HRH3
SCHEMBL28910434 0.80 CES2 (0.44) CES2CES1SMN1; SMN2ERN1
SCHEMBL20646080 0.79 CES2 (0.44) CES2CES1CYP2C19HPGDRAB9A
SCHEMBL30955355 0.78 CES2 (0.41) CES2CES1CYP2C19
SCHEMBL20645828 0.78 CES2 (0.41) CES2CES1CYP2C19
SCHEMBL9650347 0.77 CES2 (0.35) CES2CES1CYP2C19
SCHEMBL28909660 0.74
SCHEMBL28910421 0.74 CES2 (0.45) CES2CES1ERN1
SCHEMBL1971815 0.73 LMNA (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3652178-A1 BICYCLIC KETONE COMPOUNDS AND METHODS OF USE THEREOF H. Hoffnabb-La Roche Ag (CH) 2020-05-20 EP disclosed
WO-2019012063-A1 BICYCLIC KETONE COMPOUNDS AND METHODS OF USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2019-01-17 WO disclosed