SCHEMBL9650347

SCHEMBL9650347

C=CCC(CO)C(O)c1c(F)cccc1F

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9650911 0.82 CES2 (0.36) CES2CES1CYP2C19
SCHEMBL9715173 0.77 KRAS (0.30)
SCHEMBL20645990 0.77 CES2 (0.40) CES2CES1CYP2C19
SCHEMBL20640975 0.77 CES2 (0.40) CES2CES1CYP2C19
SCHEMBL9650174 0.74 CYP2C19 (0.49) CYP2C19
SCHEMBL9650334 0.70 GAA (0.37) CYP2C19
SCHEMBL9650292 0.69 SMN1; SMN2 (0.39) CES2CES1CYP2C19
SCHEMBL9162949 0.68 SMN1; SMN2 (0.33) CYP2C19
SCHEMBL28910421 0.68 CES2 (0.45) CES2CES1
SCHEMBL9036631 0.67 SMN1; SMN2 (0.44) CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166377-A Thromboxane A2 antagonist as coagulants or vasoconstrictors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-11-24 US disclosed
US-4745198-A CARDIOVASCULAR DISORDERS, BRONCHODILATOR AGENTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-05-17 US disclosed
EP-0094239-B1 1,3-DIOXAN-5-YLALKENOIC ACIDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-07-15 EP disclosed
US-4567197-A THORMBOXANE A2 ANTAGONISTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-01-28 US disclosed
EP-0094239-A2 1,3-Dioxan-5-ylalkenoic acids IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-11-16 EP disclosed