SCHEMBL20640992

SCHEMBL20640992

OCCC=Cc1ccccc1F

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 11/20 0.58
MAOB P27338 1/20 0.41
CYP1A2 P05177 2/20 0.40
RELA Q04206 1/20 0.40
CYP2D6 P10635 1/20 0.39
CYP1B1 Q16678 1/20 0.39
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20640946 0.85 PTGS2 (0.40) NFE2L2CYP1A2
SCHEMBL320615 0.83 NFE2L2 (0.62) NFE2L2MAOBCYP1A2RELACYP2D6
SCHEMBL4090323 0.83 NFE2L2 (0.62) NFE2L2MAOBCYP1A2RELACYP2D6
SCHEMBL20640938 0.78 NFE2L2 (0.45) NFE2L2
SCHEMBL20640997 0.77 NFE2L2 (0.52) NFE2L2
SCHEMBL15051245 0.77 NFE2L2 (0.54) NFE2L2RELA
SCHEMBL15051244 0.77 NFE2L2 (0.54) NFE2L2RELA
SCHEMBL15094203 0.76 HSD11B1 (0.50) RELA
SCHEMBL15539237 0.76 CHAT (0.44) NFE2L2MAOBCYP1A2RELACYP2D6
SCHEMBL5319574 0.76 CHAT (0.44) NFE2L2MAOBCYP1A2RELACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704097-A1 BICYCLIC SULFONES AND SULFOXIDES AND METHODS OF USE THEREOF F. Hoffmann-La Roche AG (CH) 2020-09-09 EP disclosed
EP-3652178-A1 BICYCLIC KETONE COMPOUNDS AND METHODS OF USE THEREOF H. Hoffnabb-La Roche Ag (CH) 2020-05-20 EP disclosed
WO-2019012063-A1 BICYCLIC KETONE COMPOUNDS AND METHODS OF USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2019-01-17 WO disclosed