SCHEMBL20645822

SCHEMBL20645822

CON(C)C(=O)c1nc2n(n1)CCC2

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.33
SLC6A3 Q01959 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20228866 0.84 RIPK1 (0.44) RIPK1ALDH1A1SMN1; SMN2
SCHEMBL20645808 0.76 MAPK1 (0.36) RIPK1ALDH1A1SMN1; SMN2
SCHEMBL19659321 0.74 ALDH1A1 (0.33) RIPK1ALDH1A1SMN1; SMN2
SCHEMBL23256256 0.73 HTT (0.35) SMN1; SMN2
SCHEMBL20645939 0.72 RIPK1 (0.44) RIPK1SMN1; SMN2
SCHEMBL20645899 0.72 RIPK1 (0.36) RIPK1SMN1; SMN2
SCHEMBL20645803 0.72 POLB (0.46) ALDH1A1
SCHEMBL20228736 0.71 RIPK1 (0.35) RIPK1ALDH1A1SMN1; SMN2
SCHEMBL20645767 0.71 RIPK1 (0.38) RIPK1SMN1; SMN2
SCHEMBL20645884 0.70 RIPK1 (0.39) RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3652178-B1 BICYCLIC KETONE COMPOUNDS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2024-01-24 EP disclosed
WO-2019012063-A1 BICYCLIC KETONE COMPOUNDS AND METHODS OF USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2019-01-17 WO disclosed