SCHEMBL20649084

SCHEMBL20649084

CC1(C)Cc2cnc(N)nc2-c2[nH]nc(C(=O)NC3NC(CN4CCC(N5CCCCC5)CC4)=CS3)c21

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 2/20 0.35
CDK2 P24941 4/20 0.32
AURKA O14965 3/20 0.32
CCNA2 P20248 1/20 0.31
CCNA1 P78396 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20649235 0.91 CDK2 (0.33) CDK2AURKACCNA2CCNA1
SCHEMBL20649268 0.89 CDK2 (0.32) CDK2AURKACCNA2CCNA1
SCHEMBL20648954 0.88 CDK2 (0.44) ACVR1CDK2AURKACCNA2CCNA1
SCHEMBL20649199 0.87 ATR (0.32)
SCHEMBL20649041 0.87 PARP1 (0.31)
SCHEMBL20649038 0.87
SCHEMBL20649146 0.85 CALCA (0.31)
SCHEMBL20648988 0.85
SCHEMBL20649387 0.85
SCHEMBL20649094 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019011715-A1 PYRAZOLO-QUINAZOLINE DERIVATIVES AS CHOLINE KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2019-01-17 WO disclosed