SCHEMBL20649199

SCHEMBL20649199

CC1(C)Cc2cnc(N)nc2-c2[nH]nc(C(=O)NC3NC(C(=O)N4CCC(N5CCCCC5)CC4)=CS3)c21

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ATR Q13535 2/20 0.32
LRRK2 Q5S007 1/20 0.32
SMYD2 Q9NRG4 1/20 0.31
L3MBTL3 Q96JM7 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20649146 0.89 CALCA (0.31)
SCHEMBL20649084 0.87 ACVR1 (0.35)
SCHEMBL20649153 0.85 LRRK2 (0.39) ATRLRRK2SMYD2L3MBTL3L3MBTL1
SCHEMBL30183348 0.85 LRRK2 (0.39) ATRLRRK2SMYD2L3MBTL3L3MBTL1
SCHEMBL30183263 0.84 LRRK2 (0.38) ATRLRRK2L3MBTL3L3MBTL1
SCHEMBL20649159 0.84 LRRK2 (0.38) ATRLRRK2L3MBTL3L3MBTL1
SCHEMBL20649191 0.84 CDK4 (0.31)
SCHEMBL20648988 0.83
SCHEMBL20649285 0.82 ATR (0.36) ATRLRRK2SMYD2L3MBTL3L3MBTL1
SCHEMBL30183031 0.82 ATR (0.36) ATRLRRK2SMYD2L3MBTL3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019011715-A1 PYRAZOLO-QUINAZOLINE DERIVATIVES AS CHOLINE KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2019-01-17 WO disclosed