SCHEMBL20649289

SCHEMBL20649289

COC(=O)c1ccc(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.47
P4HB P07237 1/20 0.43
CCR6 P51684 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
XDH P47989 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
HPGD P15428 3/20 0.37
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 4/20 0.36
HSD17B10 Q99714 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
CYP1A2 P05177 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6944749 0.93 NOTUM (0.39) NOTUMP4HBCCR6HKDC1CA12
SCHEMBL6540511 0.81 TRPA1 (0.39) NOTUMCA12CA1CA2CA7
SCHEMBL20649394 0.81 NR1H4 (0.38) CA12CA1CA2CA7XDH
SCHEMBL21876581 0.80 NR4A2 (0.39) HPGDALDH1A1HSD17B10SMN1; SMN2TSHR
SCHEMBL6592846 0.79 NOTUM (0.51) NOTUMP4HBCCR6HKDC1CA12
SCHEMBL12410847 0.78 LOXL2 (0.50) NOTUMCA12CA1CA2CA7
SCHEMBL2441663 0.78 NOTUM (0.48) NOTUMP4HBCCR6HKDC1CA12
SCHEMBL17969019 0.77 NOTUM (0.50) NOTUMCA12CA1CA2CA7
SCHEMBL18304369 0.77 MRGPRX4 (0.40) NOTUMP4HBALDH1A1MAPTGAA
SCHEMBL28847028 0.77 ABCB1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019011166-A1 MACROCYCLIC AMIDE COMPOUND, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 四川科伦博泰生物医药股份有限公司 2019-01-17 WO disclosed