SCHEMBL20649394

SCHEMBL20649394

COC(=O)c1ccc(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c(C2CC2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.38
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
CNR2 P34972 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KDM4E B2RXH2 5/20 0.36
ALDH1A1 P00352 5/20 0.36
HPGD P15428 2/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
RBP4 P02753 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20649292 0.88 CREBBP (0.36) NR1H4CNR2SLC6A4HDAC1
SCHEMBL20649289 0.81 NOTUM (0.47) KDM4EALDH1A1HPGDMAPTRAB9A
SCHEMBL22941896 0.80 CHRNB2 (0.39) NR1H4CHRNB2CHRNA4CNR2SLC6A2
SCHEMBL6540511 0.78 TRPA1 (0.39) NR1H4KDM4EALDH1A1HPGDNPC1
SCHEMBL2498155 0.77 CA12 (0.44) CHRNB2CHRNA4SLC6A2SLC6A4SLC6A3
SCHEMBL16839669 0.76 CA12 (0.42) CHRNB2CHRNA4SLC6A2SLC6A4SLC6A3
SCHEMBL2505147 0.76 CA12 (0.42) CHRNB2CHRNA4SLC6A2SLC6A4SLC6A3
SCHEMBL12410847 0.74 LOXL2 (0.50) KDM4EALDH1A1HPGDNPC1MAPT
SCHEMBL6944749 0.74 NOTUM (0.39) ALDH1A1NPC1MAPTRAB9ACA12
SCHEMBL7385091 0.73 LOXL2 (0.55) KDM4EALDH1A1HPGDMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019011166-A1 MACROCYCLIC AMIDE COMPOUND, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 四川科伦博泰生物医药股份有限公司 2019-01-17 WO disclosed