SCHEMBL2065092

SCHEMBL2065092

CCCC(O)(CN)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.47
CYP2C19 P33261 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
KIF11 P52732 4/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 1/20 0.38
ALOX12 P18054 1/20 0.38
CHRM3 P20309 1/20 0.36
KCNN4 O15554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2065923 1.00 TAAR1 (0.47) TAAR1CYP2C19CYP1A2CYP2C9KIF11
SCHEMBL2065906 1.00 TAAR1 (0.47) TAAR1CYP2C19CYP1A2CYP2C9KIF11
SCHEMBL7671955 0.89 TAAR1 (0.44) TAAR1CYP2C19CYP1A2CYP2C9KIF11
SCHEMBL9194705 0.87 CYP2C19 (0.52) CYP2C19CYP1A2CYP2C9ALDH1A1SMN1; SMN2
SCHEMBL11522604 0.87 SIGMAR1 (0.42) TAAR1CYP2C19CYP1A2CYP2C9KIF11
SCHEMBL15976484 0.85 SCN5A (0.43) TAAR1CYP2C19CYP1A2CYP2C9KIF11
Alcohol SCHEMBL1532264 0.85 TAAR1 (0.44) TAAR1CYP2C19CYP1A2CYP2C9KIF11
SCHEMBL23014014 0.83 CYP2C19 (0.48) CYP2C19CYP1A2CYP2C9ALDH1A1SMN1; SMN2
SCHEMBL1292634 0.83 TAAR1 (0.50) TAAR1CYP2C19CYP1A2CYP2C9KIF11
SCHEMBL10505123 0.83 CYP1A2 (0.56) TAAR1CYP2C19CYP1A2CYP2C9KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107921297-A Antiperspirant agent 拜尔斯道夫股份有限公司 2018-04-17 CN claimed
CN-107847769-A Antiperspirant agent 拜尔斯道夫股份有限公司 2018-03-27 CN claimed
CN-107847770-A Antiperspirant agent 拜尔斯道夫股份有限公司 2018-03-27 CN claimed
CN-107847404-A Cosmetic preparation for reducing perspiration 拜尔斯道夫股份有限公司 2018-03-27 CN claimed
CN-107847771-A Antiperspirant agent 拜尔斯道夫股份有限公司 2018-03-27 CN claimed
CN-107847403-A Cosmetic preparation for reducing perspiration 拜尔斯道夫股份有限公司 2018-03-27 CN claimed
CN-108472211-A Method for reducing perspiration 拜尔斯道夫股份有限公司 2018-08-31 CN disclosed
CN-107921297-A Antiperspirant agent 拜尔斯道夫股份有限公司 2018-04-17 CN disclosed
CN-107847769-A Antiperspirant agent 拜尔斯道夫股份有限公司 2018-03-27 CN disclosed
CN-107847770-A Antiperspirant agent 拜尔斯道夫股份有限公司 2018-03-27 CN disclosed
CN-107847404-A Cosmetic preparation for reducing perspiration 拜尔斯道夫股份有限公司 2018-03-27 CN disclosed
CN-107847771-A Antiperspirant agent 拜尔斯道夫股份有限公司 2018-03-27 CN disclosed
CN-107847403-A Cosmetic preparation for reducing perspiration 拜尔斯道夫股份有限公司 2018-03-27 CN disclosed
US-6624175-B2 4-heterocyclic substituted quinoline derivative treats disorderes associated with pathogenic neurokinin-3 receptor, such as anxiety, depression, schizophrenia, obesity, chronic pulmonary obstructive disorder or pain NEUROGEN CORPORATION 2003-09-23 US disclosed
EP-1165542-B1 4-SUBSTITUTED QUINOLINE DERIVATIVES AS NK-3 AND/OR GABA(A) RECEPTOR LIGANDS NEUROGEN CORP (US) 2003-08-20 EP disclosed
US-20020198232-A1 4-substituted quinoline derivatives NEUROGEN CORPORATION (US) 2002-12-26 US disclosed
WO-2000058303-A9 4-SUBSTITUTED QUINOLINE DERIVATIVES AS NK-3 AND/OR GABA(A) RECEPTOR LIGANDS NEUROGEN CORP (US) 2002-12-19 WO disclosed
US-6413982-B1 5-ETHYL-5-PHENYL-2-(3-METHOXY-2-PHENYLQUINOLIN-4-YL)-IMIDAZO -LINE; CENTRAL AND PERIPHERAL NERVOUS SYSTEM DISEASES AND DISORDERS; BINDS WITH HIGH AFFINITY TO NEUROKININ-3 (NK-3) AND/OR GAMMA-AMINOBUTYRIC ACID RECEPTORS; SYNERGISTIC NEUROGEN CORPORATION 2002-07-02 US disclosed
EP-1165542-A1 4-SUBSTITUTED QUINOLINE DERIVATIVES AS NK-3 AND/OR GABA(A) RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2002-01-02 EP disclosed
WO-2000058303-A1 4-SUBSTITUTED QUINOLINE DERIVATIVES AS NK-3 AND/OR GABA(A) RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2000-10-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020198232-A1 4-substituted quinoline derivatives GABRA3, GABRB3, GABRR3 TAAR1 267/4885CYP2C19 707/4885CYP1A2 451/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.