SCHEMBL20656187

SCHEMBL20656187

c1cc2c(s1)-c1c(ccc3c4c(ccc13)Cc1ccsc1-4)C2

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.33
NOS2 P35228 2/20 0.33
DRD2 P14416 1/20 0.30
DRD1 P21728 1/20 0.30
DRD4 P21917 1/20 0.30
DRD5 P21918 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL50205 0.78 NOS2 (0.41) NOS3NOS2DRD2DRD1DRD4
SCHEMBL2419709 0.73 CES1 (0.36) NOS3NOS2DRD2DRD1DRD4
SCHEMBL16256694 0.71 CES1 (0.34) NOS3NOS2DRD2DRD1DRD4
SCHEMBL12279756 0.71 CES1 (0.34) NOS3NOS2DRD2DRD1DRD4
SCHEMBL20655988 0.70 NOS3 (0.33) NOS3NOS2
SCHEMBL20260233 0.66 CYP2A6 (0.33)
SCHEMBL3290813 0.65 MAOA (0.46) DRD2DRD1DRD4DRD5DRD3
SCHEMBL5949876 0.64 NOS3 (0.33) NOS3NOS2
SCHEMBL16256695 0.64 CES1 (0.33) NOS3NOS2DRD2DRD1DRD4
SCHEMBL1820514 0.64 CES1 (0.41) NOS3NOS2DRD2DRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019011826-A1 RING CLOSURE REACTION MERCK PATENT GMBH (DE) 2019-01-17 WO disclosed