SCHEMBL20683513

SCHEMBL20683513

BCCCCC(N)(C(=O)O)[C@H]1C[C@@H](NCc2cccc3cccnc23)C1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.40
ADORA2A P29274 9/20 0.39
ADORA1 P30542 9/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2B P29275 1/20 0.39
HTR5A P47898 4/20 0.38
SIRT2 Q8IXJ6 2/20 0.36
GRM2 Q14416 1/20 0.35
GRM3 Q14832 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL894260 0.90 ARG1 (0.46) HDAC6ADORA2AADORA1ADORA3ADORA2B
SCHEMBL30169841 0.90 ARG1 (0.46) HDAC6ADORA2AADORA1ADORA3ADORA2B
SCHEMBL894261 0.90 ARG1 (0.46) HDAC6ADORA2AADORA1ADORA3ADORA2B
Hydrochloric Acid SCHEMBL895194 0.89 ARG1 (0.46) HDAC6ADORA2AADORA1ADORA3ADORA2B
Hydrochloric Acid SCHEMBL2566685 0.89 ARG1 (0.46) HDAC6ADORA2AADORA1ADORA3ADORA2B
Hydrochloric Acid SCHEMBL895195 0.89 ARG1 (0.46) HDAC6ADORA2AADORA1ADORA3ADORA2B
SCHEMBL20683408 0.81 ARG1 (0.50) HTR5A
Hydrochloric Acid SCHEMBL28256811 0.78 HTR5A (0.38) HDAC6ADORA2AADORA1ADORA3ADORA2B
SCHEMBL14897262 0.77 SLC6A2 (0.36) GRM2GRM3
SCHEMBL20683526 0.75 GRM2 (0.48) GRM2GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560978-B1 INHIBITORS OF ARGINASE AND THEIR THERAPEUTIC APPLICATIONS MARS INC (US) 2019-01-30 EP disclosed