SCHEMBL20686102

SCHEMBL20686102

Cc1ccc(C)c2c1C(=O)N(c1ccsc1C)C2=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.33
GRM1 Q13255 3/20 0.33
CASP3 P42574 1/20 0.33
TYMS P04818 1/20 0.32
AXL P30530 1/20 0.32
KDM4E B2RXH2 2/20 0.31
HPGD P15428 2/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31
HTT P42858 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
NR1H2 P55055 2/20 0.31
GRM4 Q14833 1/20 0.31
NR1H3 Q13133 1/20 0.31
ALDH1A1 P00352 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6925716 0.78 GRM1 (0.49) GRM1NR1H2NR1H3
SCHEMBL28752505 0.75 MGLL (0.48) HPGDHTTTDP1ALDH1A1
SCHEMBL28396965 0.73 CA9 (0.47) GRM1GRM4ALDH1A1HSD17B10
SCHEMBL17696374 0.71 HSD17B10 (0.53) KDM4EHPGDLMNAGAAHTT
SCHEMBL21474631 0.70 DPP4 (0.37) DPP4KDM4EHPGDTDP1NR1H2
SCHEMBL28407462 0.70 GRM1 (0.48) GRM1GRM4
SCHEMBL28398982 0.70 AR (0.49) GRM1GRM4
SCHEMBL28399876 0.68 ALDH1A1 (0.41) DPP4GRM1KDM4EHPGDLMNA
SCHEMBL21478341 0.67 MEN1 (0.38) DPP4TYMSHPGDALDH1A1
SCHEMBL21478347 0.66 MEN1 (0.39) TYMSALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3087069-B1 COMPOUNDS USEFUL AS CCR9 MODULATORS NORGINE BV (NL) 2019-01-30 EP disclosed