SCHEMBL20721895

SCHEMBL20721895

O=C(O)c1ccc(C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.59
DAO P14920 1/20 0.59
NAPRT Q6XQN6 1/20 0.59
SRD5A2 P31213 5/20 0.57
TP53 P04637 1/20 0.57
CES2 O00748 1/20 0.56
CES1 P23141 1/20 0.56
RARB P10826 1/20 0.52
RARG P13631 1/20 0.52
RXRA P19793 2/20 0.52
RXRB P28702 2/20 0.52
TRPA1 O75762 1/20 0.50
KIF11 P52732 1/20 0.49
EPHX2 P34913 1/20 0.48
NR1H4 Q96RI1 1/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA12 O43570 1/20 0.48
CA3 P07451 1/20 0.48
TYR P14679 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18896444 1.00 TSHR (0.59) TSHRDAONAPRTSRD5A2TP53
SCHEMBL2176223 0.93 TSHR (0.67) TSHRDAONAPRTSRD5A2TP53
SCHEMBL23861614 0.92 CA12 (0.64) TSHRDAONAPRTSRD5A2TP53
SCHEMBL6351953 0.88 SRD5A2 (0.65) TSHRDAONAPRTSRD5A2RXRA
SCHEMBL16772180 0.86 RXRA (0.62) TSHRSRD5A2TP53RARBRARG
SCHEMBL407595 0.84 TSHR (0.56) TSHRDAONAPRTSRD5A2TP53
SCHEMBL5311010 0.84 TSHR (0.56) TSHRDAONAPRTSRD5A2TP53
SCHEMBL27683133 0.84 ALDH1A1 (0.57) SRD5A2RXRARXRBEPHX2NR1H4
SCHEMBL23861613 0.82 TSHR (0.45) TSHRDAONAPRTSRD5A2TP53
SCHEMBL13956160 0.82 KCNN4 (0.61) TSHRDAONAPRTSRD5A2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10787576-B2 Method for the preparation of a coating comprising oligomeric alkynes ÉCOLE POLYTECHNIQUE FÉDÉRALE DE LAUSANNE (EPFL) EPFL-TTO (CH) 2020-09-29 US disclosed
US-20190048202-A1 METHOD FOR THE PREPARATION OF A COATING COMPRISING OLIGOMERIC ALKYNES ÉCOLE POLYTECHNIQUE FÉDÉRALE DE LAUSANNE (EPFL) EPFL-TTO (CH) 2019-02-14 US disclosed
CN-105051048-B 1-hydroxy-benzoxaboroles as antiparasitic agents 伊莱利利公司 2017-03-15 CN disclosed
CN-105051048-A 1-hydroxy-benzoxaboroles as antiparasitic agents LILLY CO ELI 2015-11-11 CN disclosed