SCHEMBL2073159

SCHEMBL2073159

N#Cc1c(F)cccc1NCc1cccs1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 1.00
HPGD P15428 3/20 0.42
ACHE P22303 1/20 0.41
CYP1A2 P05177 5/20 0.41
CYP3A4 P08684 5/20 0.41
CYP2D6 P10635 5/20 0.41
CYP2C19 P33261 4/20 0.41
LMNA P02545 4/20 0.41
MAPK1 P28482 3/20 0.41
HSD17B10 Q99714 3/20 0.41
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GLA P06280 1/20 0.41
ALOX15 P16050 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CLK4 Q9HAZ1 4/20 0.40
MEN1 O00255 2/20 0.40
TP53 P04637 2/20 0.40
KMT2A Q03164 2/20 0.40
KCNH3 Q9ULD8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22904299 0.76 KDM4E (0.61) KDM4EHPGDACHELMNAHSD17B10
SCHEMBL7519734 0.76 KDM4E (0.61) KDM4EHPGDCYP1A2CYP3A4CYP2D6
SCHEMBL27393494 0.73 KDM4E (0.57) KDM4EHPGDACHECYP1A2HSD17B10
SCHEMBL1154871 0.71 KDM4E (0.56) KDM4EHPGDLMNAHSD17B10ALDH1A1
SCHEMBL12956699 0.71 KDM4E (0.55) KDM4EHPGDACHECYP1A2LMNA
SCHEMBL25057053 0.70 KDM4E (0.54) KDM4EHPGDACHECYP1A2HSD17B10
SCHEMBL2074476 0.69 HPGD (0.60) KDM4EHPGDCYP1A2CYP3A4CYP2D6
SCHEMBL6798736 0.68 L3MBTL1 (0.63) KDM4EHPGDCYP1A2CYP3A4CYP2D6
SCHEMBL933760 0.68 CYP1A2 (0.57) KDM4EHPGDCYP1A2CYP3A4CYP2D6
SCHEMBL5783945 0.68 KDM4E (0.51) KDM4EHPGDACHELMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7863444-B2 4-aminopyrrolopyrimidines as kinase inhibitors ABBOTT LABORATORIES (US) 2011-01-04 US disclosed