SCHEMBL20734845

SCHEMBL20734845

CC(C)CC1NC(=O)C=C1OCc1cccc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.39
CNR1 P21554 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
PARP10 Q53GL7 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37
GAA P10253 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PIN1 Q13526 1/20 0.37
FFAR1 O14842 1/20 0.36
AKR1B1 P15121 1/20 0.36
BCHE P06276 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PARP15 Q460N3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20734844 1.00 CNR2 (0.39) CNR2CNR1MEN1KMT2APARP10
SCHEMBL20734837 0.82 L3MBTL1 (0.42) CNR2CNR1MEN1KMT2APARP10
SCHEMBL20734964 0.81 CNR1 (0.38) CNR2CNR1MEN1KMT2APARP10
SCHEMBL20734943 0.81 CNR1 (0.38) CNR2CNR1MEN1KMT2APARP10
SCHEMBL20734917 0.79 AKR1B1 (0.42) MEN1KMT2APARP10ALDH1A1MAPT
SCHEMBL20734918 0.79 AKR1B1 (0.42) MEN1KMT2APARP10ALDH1A1MAPT
SCHEMBL24333190 0.75 CYP2D6 (0.36) CNR2CNR1MEN1KMT2APARP10
SCHEMBL21927113 0.73 PRCP (0.31)
SCHEMBL20734816 0.73 MAOB (0.36) MEN1KMT2AHPGD
SCHEMBL20734815 0.73 MAOB (0.36) MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019029273-A1 4-OXO-ALKYLATED TETRAMIC ACID COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 北京卓凯生物技术有限公司 2019-02-14 WO disclosed
WO-2019029274-A1 4-OXO-ALKYLATED TETRAMIC ACID COMPOUND AND PREPARATION METHOD THEREFOR 北京卓凯生物技术有限公司 2019-02-14 WO disclosed