SCHEMBL20748375

SCHEMBL20748375

COOCOCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.58
IDO1 P14902 1/20 0.43
AGXT P21549 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CA1 P00915 4/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
MAOB P27338 1/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
TACR1 P25103 2/20 0.39
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL434644 0.84 TSHR (0.61) TSHRIDO1AGXTTDP1L3MBTL1
SCHEMBL6832294 0.82 TSHR (0.64) TSHRIDO1AGXTALDH1A1CA1
SCHEMBL3127292 0.82 TSHR (0.64) TSHRIDO1AGXTTDP1L3MBTL1
SCHEMBL26656 0.81 TSHR (0.55) TSHRIDO1AGXTTDP1L3MBTL1
SCHEMBL223907 0.81 TSHR (0.78) TSHRIDO1AGXTALDH1A1CA1
SCHEMBL70291 0.79 TSHR (0.74) TSHRIDO1AGXTTDP1L3MBTL1
SCHEMBL53267 0.79 TSHR (0.74) TSHRIDO1AGXTTDP1L3MBTL1
SCHEMBL434643 0.78 TSHR (0.58) TSHRIDO1AGXTTDP1L3MBTL1
SCHEMBL5353833 0.76 TSHR (0.61) TSHRIDO1AGXTTDP1L3MBTL1
SCHEMBL5311581 0.75 TSHR (1.00) TSHRIDO1AGXTALDH1A1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2928869-B1 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS CHIESI FARM SPA (IT) 2019-02-20 EP disclosed