SCHEMBL20748604

SCHEMBL20748604

C=C/C=C\C(C)=C/C(=C)c1cc(C(=O)NC)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.41
NPC1 O15118 1/20 0.38
DOT1L Q8TEK3 1/20 0.37
KMT2A Q03164 1/20 0.36
CREBBP Q92793 1/20 0.35
KDM4E B2RXH2 2/20 0.33
HTT P42858 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
SMYD3 Q9H7B4 2/20 0.32
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
ALDH1A1 P00352 2/20 0.31
GAA P10253 1/20 0.31
AKR1C3 P42330 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
BAZ2B Q9UIF8 1/20 0.30
BAZ2A Q9UIF9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20748511 0.86 NOTUM (0.39) NPC1SMYD3GAA
SCHEMBL20748490 0.81 ALDH1A1 (0.33) ALDH1A1BAZ2BBAZ2A
SCHEMBL20748611 0.73 MEN1 (0.39) KMT2AHTTALDH1A1GAAL3MBTL1
SCHEMBL20748481 0.72 NOTUM (0.41) BRD4NPC1SMYD3GAABAZ2B
SCHEMBL20748619 0.71 EGLN1 (0.35) BRD4KMT2AHTTSMYD3ALDH1A1
SCHEMBL20748646 0.69 ALDH1A1 (0.36) KMT2AKDM4EHTTALDH1A1GAA
SCHEMBL20748517 0.68
SCHEMBL18410439 0.63 NOTUM (0.59) BRD4NPC1DOT1LKMT2ACREBBP
SCHEMBL18236154 0.60 BRD4 (0.46) BRD4NPC1DOT1LKMT2ACREBBP
SCHEMBL20748631 0.60

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2473501-B1 COMPOUNDS AS TYROSINE KINASE MODULATORS ALLERGAN INC (US) 2019-02-20 EP disclosed