SCHEMBL20748619

SCHEMBL20748619

C=C(/C=C(C)\C=C/C)c1cc(C(=O)NCCC(=O)O)c[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 3/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
ITGB3 P05106 2/20 0.33
ITGA2B P08514 2/20 0.33
BRD4 O60885 1/20 0.33
FABP4 P15090 1/20 0.33
MAPK1 P28482 1/20 0.32
NME4 O00746 2/20 0.32
GCDH Q92947 2/20 0.32
SIRT5 Q9NXA8 2/20 0.32
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
CHRM1 P11229 1/20 0.32
ADORA2A P29274 1/20 0.32
AVPR2 P30518 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20748646 0.83 ALDH1A1 (0.36) MEN1KMT2AALDH1A1HTTL3MBTL1
SCHEMBL20748481 0.81 NOTUM (0.41) BRD4TDP1SMYD3
SCHEMBL20748517 0.75
SCHEMBL29953684 0.73 SMYD3 (0.51) EGLN1MEN1KMT2AALDH1A1BRD4
SCHEMBL20748611 0.72 MEN1 (0.39) MEN1KMT2AALDH1A1FABP4MAPK1
SCHEMBL20748604 0.71 BRD4 (0.41) KMT2AALDH1A1BRD4HTTL3MBTL1
SCHEMBL20748511 0.69 NOTUM (0.39) TDP1SMYD3
SCHEMBL29953018 0.66 MEN1 (0.52) MEN1KMT2AALDH1A1FABP4MAPK1
SCHEMBL29958499 0.64 MAPK1 (0.54) MEN1KMT2AALDH1A1ITGB3ITGA2B
SCHEMBL394245 0.64 FABP4 (0.59) ALDH1A1CA1CA2ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2473501-B1 COMPOUNDS AS TYROSINE KINASE MODULATORS ALLERGAN INC (US) 2019-02-20 EP disclosed