SCHEMBL20749362

SCHEMBL20749362

CCCSNc1cc(F)c(F)c(C(=O)c2ccc3ncc(C)nc3c2)c1F

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.34
KDM4E B2RXH2 3/20 0.34
RAB9A P51151 2/20 0.34
HTT P42858 1/20 0.34
BRAF P15056 3/20 0.33
MGLL Q99685 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KCNQ3 O43525 1/20 0.30
KCNQ2 O43526 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
VNN1 O95497 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC2 Q92769 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20749378 0.85 CDK6 (0.41) BRAFKCNQ3KCNQ2HDAC3HDAC2
SCHEMBL14716226 0.82 BRAF (0.52) BRAF
SCHEMBL14829805 0.78 HSD17B14 (0.39) NPC1RAB9AMGLLTDP1
SCHEMBL18627722 0.77 RAB9A (0.40) NPC1KDM4ERAB9AHTTBRAF
SCHEMBL18627635 0.76 CDK6 (0.43) BRAFKCNQ3KCNQ2HDAC3HDAC2
SCHEMBL14716059 0.76 SLC40A1 (0.43) BRAFMEN1KMT2AALDH1A1
SCHEMBL14716241 0.76 BRAF (0.47) BRAF
SCHEMBL14716257 0.74 BRAF (0.57) BRAF
SCHEMBL14716062 0.74 CYP3A4 (0.47) BRAFSMN1; SMN2HDAC3HDAC2
SCHEMBL14716086 0.73 BRAF (0.51) BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2747767-B1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS NEUPHARMA INC (US) 2019-02-20 EP disclosed