SCHEMBL20765451

SCHEMBL20765451

COc1ccc(OCCCc2nc3cc(C(=O)N4CCN(Cc5ccccc5OC)CC4)ccc3[nH]2)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.54
USP2 O75604 2/20 0.54
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 2/20 0.52
HTT P42858 1/20 0.52
DRD2 P14416 7/20 0.51
DRD3 P35462 5/20 0.51
NPC1 O15118 1/20 0.49
CYP3A4 P08684 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.47
KCNA5 P22460 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20765595 0.85 DRD3 (0.51) ALDH1A1DRD2DRD3KCNA5MAPT
SCHEMBL20765784 0.85 KDM4E (0.48) ALDH1A1KDM4EHTTDRD2DRD3
SCHEMBL20765619 0.78 ALDH1A1 (0.40) ALDH1A1DRD2DRD3MAPT
SCHEMBL20765618 0.78 ALDH1A1 (0.40) ALDH1A1DRD2DRD3MAPT
SCHEMBL20765555 0.78 ALDH1A1 (0.66) CYP2D6USP2ALDH1A1KDM4EHTT
SCHEMBL20765612 0.74 ALDH1A1 (0.56) ALDH1A1KDM4EHTTNPC1
SCHEMBL20765771 0.73 ALDH1A1 (0.59) CYP2D6USP2ALDH1A1KDM4EHTT
SCHEMBL20765593 0.73 KDM4E (0.48) ALDH1A1KDM4EHTTDRD2DRD3
SCHEMBL19970844 0.70 LMNA (0.46) ALDH1A1KDM4EHTTNPC1SMN1; SMN2
SCHEMBL20774925 0.70 ALDH1A1 (0.52) ALDH1A1KDM4EHTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO claimed