SCHEMBL20765495

SCHEMBL20765495

N#Cc1ccccc1CN1CCN(C(=O)c2ccc3nc(-c4ccccc4)[nH]c3c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.56
BCHE P06276 2/20 0.51
ACHE P22303 2/20 0.51
CHEK2 O96017 7/20 0.49
ACACB O00763 2/20 0.47
ACACA Q13085 1/20 0.47
HDAC6 Q9UBN7 4/20 0.47
HDAC3 O15379 2/20 0.47
HDAC1 Q13547 2/20 0.47
HDAC8 Q9BY41 2/20 0.47
HDAC2 Q92769 1/20 0.47
HPGD P15428 1/20 0.46
MAPK14 Q16539 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20765497 0.87 MGLL (0.58) MGLLBCHEACHECHEK2ACACB
SCHEMBL20765786 0.83 BCHE (0.55) MGLLBCHEACHECHEK2ACACB
SCHEMBL20765523 0.82 MGLL (0.58) MGLLBCHEACHECHEK2ACACB
SCHEMBL20765616 0.81 KDM4E (0.52) MGLLBCHEACHECHEK2HDAC6
SCHEMBL20765511 0.79 ACACB (0.59) MGLLACACBHPGD
SCHEMBL20765715 0.79 ALDH1A1 (0.56) MGLLCHEK2HPGDMAPK14
SCHEMBL20782579 0.79 ALDH1A1 (0.55) MGLLBCHEACHEHPGDMAPK14
SCHEMBL19970807 0.79 ACACB (0.62) MGLLBCHEACHECHEK2ACACB
SCHEMBL21843704 0.79 HPGD (0.70) MGLLCHEK2ACACBACACAHDAC6
SCHEMBL16619560 0.78 MGLL (0.65) MGLLCHEK2ACACBACACAHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO claimed
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO disclosed