SCHEMBL20765710

SCHEMBL20765710

O=C(c1ccc2[nH]c(-c3ccccc3)nc2c1)N1CCN(Cc2ccc(F)cc2F)CC1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.48
MGLL Q99685 2/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 5/20 0.46
GAA P10253 1/20 0.46
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MAPK14 Q16539 2/20 0.45
HTT P42858 1/20 0.44
BRD4 O60885 1/20 0.43
NPC1 O15118 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
GRIN2B Q13224 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20782579 0.92 ALDH1A1 (0.55) HPGDMGLLKDM4EALDH1A1GAA
SCHEMBL20765467 0.85 ALDH1A1 (0.52) HPGDMGLLKDM4EALDH1A1GAA
SCHEMBL20765715 0.84 ALDH1A1 (0.56) HPGDMGLLKDM4EALDH1A1GAA
SCHEMBL20765497 0.84 MGLL (0.58) HPGDMGLLKDM4EALDH1A1MEN1
SCHEMBL20765580 0.83 KDM4E (0.50) HPGDKDM4EALDH1A1MEN1LMNA
SCHEMBL20765518 0.82 KDM4E (0.47) HPGDMGLLKDM4EALDH1A1MEN1
SCHEMBL20765510 0.82 ALDH1A1 (0.48) HPGDKDM4EALDH1A1GAAMEN1
SCHEMBL20765528 0.81 ALDH1A1 (0.50) HPGDMGLLKDM4EALDH1A1GAA
SCHEMBL20765547 0.81 MAPK14 (0.55) HPGDMGLLKDM4EALDH1A1MEN1
SCHEMBL20774945 0.81 MAPK14 (0.55) HPGDMGLLALDH1A1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO claimed
WO-2019038683-A1 COMPOUNDS TARGETING TANDEM BRCT DOMAINS OF BRCA1, COMPOSITIONS AND METHODS THEREOF INSTITUTE FOR STEM CELL BIOLOGY AND REGENERATIVE MEDICINE (IN) 2019-02-28 WO disclosed