SCHEMBL20767744

SCHEMBL20767744

CC(NC(=O)OCc1ccccc1)C(O[Si](C)(C)C(C)(C)C)C(C)NC(=O)OC(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.54
ATM Q13315 3/20 0.50
MAPT P10636 2/20 0.50
PPARA Q07869 1/20 0.46
CTSK P43235 4/20 0.46
POLB P06746 1/20 0.45
CTSS P25774 2/20 0.43
CTSL P07711 2/20 0.43
KLK7 P49862 1/20 0.43
KLK5 Q9Y337 1/20 0.43
CTSB P07858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18163524 1.00 SYK (0.54) SYKATMMAPTPPARACTSK
SCHEMBL16823456 1.00 SYK (0.54) SYKATMMAPTPPARACTSK
SCHEMBL18143168 1.00 SYK (0.54) SYKATMMAPTPPARACTSK
SCHEMBL16823454 1.00 SYK (0.54) SYKATMMAPTPPARACTSK
SCHEMBL18157219 0.90 ATM (0.53) SYKATMCTSKCTSSCTSL
SCHEMBL19812740 0.82 SYK (0.61) SYKATMMAPTPPARACTSK
SCHEMBL16824022 0.82 SYK (0.61) SYKATMMAPTPPARACTSK
SCHEMBL18143207 0.82 SYK (0.61) SYKATMMAPTPPARACTSK
SCHEMBL16824023 0.82 SYK (0.61) SYKATMMAPTPPARACTSK
SCHEMBL6381541 0.81 SYK (0.60) SYKATMMAPTPPARACTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10221146-B2 Tetrahydronaphthyridine, benzoxazine, aza-benzoxazine and related bicyclic compounds for inhibition of RORgamma activity and the treatment of disease LYCERA CORPORATION (US) 2019-03-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10221146-B2 Tetrahydronaphthyridine, benzoxazine, aza-benzoxazine and related bicyclic compounds for inhibition of RORgamma activity and the treatment of disease RORB, RORA, RORC SYK 2404/4885ATM 4865/4885MAPT 3559/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.