SCHEMBL20769718

SCHEMBL20769718

O=C(O)Cc1nn(Cc2ccccc2Cl)c2ccc(Cl)cc12

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 16/20 0.62
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
TSHR P16473 1/20 0.55
PMP22 Q01453 1/20 0.55
HIF1A Q16665 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
PTGDR2 Q9Y5Y4 1/20 0.52
CCR2 P41597 1/20 0.48
SLC22A12 Q96S37 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3247322 0.80 AKR1B1 (0.57) AKR1B1PTGDR2
SCHEMBL9321434 0.80 AKR1B1 (0.67) AKR1B1PTGDR2
SCHEMBL9322563 0.79 AKR1B1 (0.66) AKR1B1
SCHEMBL9218891 0.78 AKR1B1 (0.66) AKR1B1CYP1A2CYP2C9PTGDR2
SCHEMBL9322351 0.77 AKR1B1 (1.00) AKR1B1
SCHEMBL9323846 0.77 AKR1B1 (1.00) AKR1B1
SCHEMBL20769651 0.76 ALDH1A1 (0.60) CYP2C9NPSR1CCR2SLC22A12
SCHEMBL8038414 0.75 AKR1B1 (0.53) AKR1B1
SCHEMBL9323969 0.74 AKR1B1 (0.51) AKR1B1PTGDR2
SCHEMBL5317956 0.73 AKR1B1 (0.56) AKR1B1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019046668-A1 AMIDE SUBSTITUTED THIAZOLES AS PROTEIN SECRETION INHIBITORS KEZAR LIFE SCIENCES (US) 2019-03-07 WO disclosed