Bropirimine

Bropirimine

SCHEMBL20769828

Nc1nc(=O)c(Br)c(-c2ccccc2)[nH]1.Nc1nc(=O)c(Br)c(-c2ccccc2)[nH]1

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 8/20 0.57
FGFR1 P11362 1/20 0.43
FGFR2 P21802 1/20 0.43
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
KDM4E B2RXH2 1/20 0.42
PLA2G10 O15496 1/20 0.42
GAA P10253 1/20 0.42
HSD17B10 Q99714 1/20 0.42
QTRT1 Q9BXR0 1/20 0.42
MASP2 O00187 1/20 0.41
NOS1 P29475 1/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
MAPK13 O15264 1/20 0.38
GCGR P47871 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bropirimine SCHEMBL4058 1.00 XDH (0.57) XDHFGFR1FGFR2ALDH1A1HPGD
Bropirimine SCHEMBL5271073 0.82 XDH (0.41) XDHFGFR1FGFR2ALDH1A1HPGD
SCHEMBL19665218 0.81 MAPK13 (0.54) XDHALDH1A1HPGDKDM4EPLA2G10
SCHEMBL8995841 0.81 XDH (0.49) XDHFGFR1FGFR2ALDH1A1HPGD
SCHEMBL15928125 0.79 KDM4E (0.56) XDHALDH1A1HPGDKDM4EPLA2G10
SCHEMBL19733297 0.76 XDH (0.60) XDHALDH1A1HPGDADORA2AADORA1
SCHEMBL5383500 0.74 MAPK13 (0.60) ALDH1A1HPGDHSD17B10MAPTMAPK13
Bropirimine SCHEMBL509127 0.72 XDH (1.00) XDHFGFR1FGFR2ALDH1A1HPGD
SCHEMBL725362 0.72 KDM4E (0.60) XDHALDH1A1HPGDKDM4EGAA
SCHEMBL31683723 0.71 XDH (0.46) XDHFGFR1FGFR2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3675838-A1 LYMPHATIC SYSTEM-DIRECTING LIPID PRODRUGS Puretecch LYT, Inc. (US) 2020-07-08 EP disclosed
CN-109988240-A Anti- GPC-3 antibody and application thereof 安源生物科技(上海)有限公司 2019-07-09 CN disclosed
WO-2019046491-A1 LYMPHATIC SYSTEM-DIRECTING LIPID PRODRUGS ARIYA THERAPEUTICS, INC. (US) 2019-03-07 WO disclosed