SCHEMBL20780879

SCHEMBL20780879

C=C(O)c1nc(C)ccc1-c1ncc(C(F)(F)F)cn1

nearest known ligand 0.43

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 16/20 0.43
HCRTR2 O43614 11/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3385652 0.86 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL30775081 0.86 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL20781141 0.83 HCRTR1 (0.38) HCRTR1HCRTR2
SCHEMBL7901595 0.76 HCRTR1 (0.37) HCRTR1HCRTR2
SCHEMBL30775065 0.72 ALDH1A1 (0.39) HCRTR1HCRTR2
SCHEMBL3388543 0.72 ALDH1A1 (0.39) HCRTR1HCRTR2
SCHEMBL3387269 0.69 HCRTR2 (0.46) HCRTR1HCRTR2
SCHEMBL27831836 0.68 HDAC4 (0.45)
SCHEMBL30775053 0.68 HCRTR2 (0.42) HCRTR1HCRTR2
SCHEMBL2471955 0.68 HCRTR2 (0.42) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019043407-A1 SUBSTITUTED 2-AZABICYCLO[3.1.1]HEPTANE AND 2-AZABICYCLO[3.2.1]OCTANE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS CHRONOS THERAPEUTICS LIMITED (GB) 2019-03-07 WO disclosed