SCHEMBL7901595

SCHEMBL7901595

Cc1ccc(-c2ncc(C(F)(F)F)cn2)c(N)n1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 9/20 0.37
HCRTR2 O43614 8/20 0.37
MBOAT4 Q96T53 1/20 0.33
HDAC4 P56524 1/20 0.33
HEXA P06865 1/20 0.33
HEXB P07686 1/20 0.33
POLB P06746 1/20 0.33
PDE2A O00408 1/20 0.33
NFKBIA P25963 1/20 0.33
RELA Q04206 1/20 0.33
MAP4K4 O95819 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30775065 0.77 ALDH1A1 (0.39) HCRTR1HCRTR2
SCHEMBL3388543 0.77 ALDH1A1 (0.39) HCRTR1HCRTR2
SCHEMBL3385652 0.76 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL30775081 0.76 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL20780879 0.76 HCRTR1 (0.43) HCRTR1HCRTR2
SCHEMBL13637232 0.75 NOS3 (0.42) HCRTR1HCRTR2POLB
SCHEMBL26521057 0.70 CCR1 (0.50)
SCHEMBL27831836 0.69 HDAC4 (0.45) HDAC4
SCHEMBL15230506 0.68 METAP2 (0.59)
SCHEMBL15539272 0.67 MBOAT4 (0.41) MBOAT4HEXAHEXBPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063663-A1 N-{[(IR,4S,6R-3-(2-PYRIDINYLCARBONYL)-3-AZABICYCLO [4.1.0]HEPT-4-YL] METHYL}-2-HETEROARYLAMINE DERIVATIVES AND USES THEREOF GLAXO GROUP LIMITED (GB) 2010-06-10 WO disclosed