SCHEMBL20780901

SCHEMBL20780901

C=C(O)c1nc(C)sc1-c1ccc(F)cc1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.47
HCRTR1 O43613 14/20 0.46
HCRTR2 O43614 14/20 0.46
ALOX5 P09917 2/20 0.44
PDPK1 O15530 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL270942 0.84 HCRTR1 (0.51) PTGS2HCRTR1HCRTR2ALOX5
SCHEMBL27854218 0.82 HCRTR1 (0.52) PTGS2HCRTR1HCRTR2PDPK1
SCHEMBL20780900 0.81 ALOX5 (0.41) PTGS2HCRTR1HCRTR2ALOX5
SCHEMBL20780957 0.79 HCRTR1 (0.41) PTGS2HCRTR1HCRTR2ALOX5
SCHEMBL1257080 0.79 HCRTR1 (0.50) PTGS2HCRTR1HCRTR2PDPK1
SCHEMBL271104 0.77 KDM4E (0.53) PTGS2HCRTR1HCRTR2
SCHEMBL14705611 0.76 KDM4E (0.45) PTGS2
SCHEMBL320589 0.75 PTGS2 (0.54) PTGS2HCRTR1HCRTR2ALOX5PDPK1
SCHEMBL21615547 0.73 PTGS2 (0.51) PTGS2HCRTR1HCRTR2ALOX5PDPK1
SCHEMBL28786381 0.71 KDM4E (0.49) PTGS2HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019043407-A1 SUBSTITUTED 2-AZABICYCLO[3.1.1]HEPTANE AND 2-AZABICYCLO[3.2.1]OCTANE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS CHRONOS THERAPEUTICS LIMITED (GB) 2019-03-07 WO disclosed