SCHEMBL20780957

SCHEMBL20780957

C=C(O)c1nc(C)sc1-c1ccc(C)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.41
HCRTR2 O43614 4/20 0.41
ALOX5 P09917 1/20 0.39
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PI4KA P42356 1/20 0.38
PIK3CG P48736 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
HPGDS O60760 1/20 0.38
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
PTGS2 P35354 2/20 0.35
TDO2 P48775 1/20 0.35
HSD17B10 Q99714 3/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
PDE10A Q9Y233 2/20 0.33
POLQ O75417 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20773621 0.86 HCRTR1 (0.45) HCRTR1HCRTR2ALOX5PIK3CDPIK3CA
SCHEMBL20780901 0.79 PTGS2 (0.47) HCRTR1HCRTR2ALOX5PTGS2
SCHEMBL20781037 0.78 JAK2 (0.45) ALOX5PIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL20773528 0.77 ALDH1A1 (0.46) HCRTR1HCRTR2NPC1
SCHEMBL20780900 0.77 ALOX5 (0.41) HCRTR1HCRTR2ALOX5PTGS2TSHR
SCHEMBL1968622 0.70 HCRTR1 (0.51) HCRTR1HCRTR2PIK3CDPIK3CAPIK3CB
SCHEMBL676678 0.66 HPGDS (0.56) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL13750611 0.66 HSD17B10 (0.48) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL268643 0.66 KDM4E (0.49) HCRTR1HCRTR2ALOX5RAB9AHSD17B10
SCHEMBL2405110 0.65 HPGDS (0.43) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019043407-A1 SUBSTITUTED 2-AZABICYCLO[3.1.1]HEPTANE AND 2-AZABICYCLO[3.2.1]OCTANE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS CHRONOS THERAPEUTICS LIMITED (GB) 2019-03-07 WO disclosed