SCHEMBL20782852

SCHEMBL20782852

COc1ccc2c(-c3ccc(CN[S+](N)[O-])s3)ccnc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP3 O14638 1/20 0.45
ENPP1 P22413 1/20 0.45
HTR1A P08908 3/20 0.43
ADRA1D P25100 3/20 0.43
ADRA1A P35348 3/20 0.43
ADRA1B P35368 3/20 0.43
FERMT2 Q96AC1 1/20 0.42
TLR8 Q9NR97 3/20 0.41
KCNH2 Q12809 1/20 0.38
GRM4 Q14833 1/20 0.38
GAK O14976 1/20 0.36
RIPK2 O43353 1/20 0.36
COQ8A Q8NI60 1/20 0.36
NLK Q9UBE8 1/20 0.36
AKT1 P31749 1/20 0.35
MET P08581 5/20 0.35
CSF1R P07333 1/20 0.35
PDGFRB P09619 1/20 0.35
KDR P35968 1/20 0.35
EGFR P00533 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22407387 0.81 ENPP1 (0.66) ENPP3ENPP1HTR1AADRA1DADRA1A
SCHEMBL22407385 0.81 ENPP3 (0.47) ENPP3ENPP1HTR1AADRA1DADRA1A
SCHEMBL22436143 0.64 ENPP3 (0.67) ENPP3ENPP1HTR1AADRA1DADRA1A
SCHEMBL9159084 0.64 GRM4 (0.67) ENPP3ENPP1HTR1AADRA1DADRA1A
SCHEMBL9139295 0.63 TLR8 (0.59) ENPP3ENPP1HTR1AADRA1DADRA1A
Hydrochloric Acid SCHEMBL20771109 0.63 ENPP3 (0.66) ENPP3ENPP1HTR1AADRA1DADRA1A
SCHEMBL3841526 0.63 HTR1A (0.58) ENPP3ENPP1HTR1AADRA1DADRA1A
SCHEMBL28436096 0.62 TLR8 (0.61) ENPP3ENPP1HTR1AADRA1DADRA1A
SCHEMBL25620299 0.62 MET (0.52) HTR1AADRA1DADRA1AADRA1BFERMT2
SCHEMBL20770893 0.62 ENPP1 (1.00) ENPP3ENPP1HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019046778-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE 1 (ENPP-1) INHIBITORS AND USES THEREOF MAVUPHARMA, INC. (US) 2019-03-07 WO disclosed