SCHEMBL20804153

SCHEMBL20804153

Cc1cccc(CN(C)C(=O)/C=C\C=O)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.48
HSD17B2 P37059 3/20 0.44
HSD17B1 P14061 2/20 0.44
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
ACHE P22303 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GPR52 Q9Y2T5 1/20 0.40
TAS2R14 Q9NYV8 1/20 0.40
AOC3 Q16853 2/20 0.39
CTBP2 P56545 1/20 0.38
POLB P06746 2/20 0.38
LIMK1 P53667 1/20 0.38
LIMK2 P53671 1/20 0.38
HPGD P15428 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PLAU P00749 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22018330 0.83 NPC1 (0.54) MEN1KMT2AHPGD
SCHEMBL20804235 0.82 HSP90AA1 (0.43) HSP90AA1POLB
SCHEMBL13114705 0.77 HSP90AA1 (0.56) HSP90AA1HSD17B2HSD17B1ACHEMEN1
SCHEMBL18773897 0.76 KMT2A (0.69) HSP90AA1HSD17B2HSD17B1MEN1KMT2A
SCHEMBL20804162 0.75 HDAC1 (0.33)
SCHEMBL14524623 0.74 HSP90AA1 (0.53) HSP90AA1HSD17B2HSD17B1MEN1KMT2A
SCHEMBL24011318 0.73 HSP90AA1 (0.52) HSP90AA1HSD17B2HSD17B1SLC6A2SLC6A4
SCHEMBL13887741 0.73 RIPK1 (0.54) HSP90AA1HSD17B2HSD17B1ACHEMEN1
SCHEMBL16127892 0.73 HSP90AA1 (0.52) HSP90AA1HSD17B2HSD17B1ACHEMEN1
SCHEMBL19577474 0.72 SMN1; SMN2 (0.56) HSP90AA1ACHEMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3089962-B1 RADIOIODINATED COMPOUNDS NUTECH VENTURES (US) 2019-03-13 EP disclosed