SCHEMBL20805366

SCHEMBL20805366

Cc1ccc(-c2ccc3c(c2)C(C)(C)OC32CCCC2)nc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.40
CCR1 P32246 1/20 0.39
CCR5 P51681 1/20 0.39
CCR8 P51685 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
GRIA2 P42262 1/20 0.38
CYP3A4 P08684 1/20 0.36
CYP2A6 P11509 1/20 0.36
ALOX5AP P20292 2/20 0.34
METAP2 P50579 1/20 0.34
BACE1 P56817 2/20 0.33
KDM1A O60341 1/20 0.33
MERTK Q12866 1/20 0.32
PTGS2 P35354 2/20 0.32
P2RX3 P56373 2/20 0.31
P2RX2 Q9UBL9 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17486214 0.86 BACE1 (0.32) ALOX5APBACE1
SCHEMBL17486187 0.81 DGAT1 (0.46)
SCHEMBL17486140 0.77 RARA (0.37) ALOX5AP
SCHEMBL18790585 0.76 CCR1 (0.47) P2RX7CCR1CCR5CCR8HDAC6
SCHEMBL22202855 0.72 PGR (0.30)
SCHEMBL22202500 0.70 PDE7A (0.31)
SCHEMBL12721334 0.70 CCR1 (0.47) P2RX7CCR1CCR5CCR8HDAC6
SCHEMBL15614861 0.69 BACE2 (0.33) BACE1KDM1A
SCHEMBL17486216 0.69 MAPK1 (0.37) BACE1PTGS2
SCHEMBL22202605 0.68 PGR (0.35) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3174890-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-03-13 EP disclosed