SCHEMBL20830463

SCHEMBL20830463

COc1ccc2c3c(ccnc13)C(=O)N(c1ccc(C)cc1)C2=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.56
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 7/20 0.47
UGCG Q16739 1/20 0.44
NPC1 O15118 2/20 0.43
HSD17B10 Q99714 2/20 0.43
TSHR P16473 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
NR1H3 Q13133 2/20 0.42
NR1H2 P55055 1/20 0.42
POLB P06746 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4E B2RXH2 2/20 0.41
CA9 Q16790 2/20 0.41
HPGD P15428 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20830396 0.88 ALDH1A1 (0.56) RAB9AMEN1KMT2AALDH1A1UGCG
SCHEMBL20830481 0.81 ALDH1A1 (0.49) RAB9AMEN1KMT2AALDH1A1NPC1
SCHEMBL13400250 0.80 RAB9A (0.60) RAB9AMEN1KMT2AALDH1A1NPC1
SCHEMBL20735081 0.75 RAB9A (0.56) RAB9AMEN1KMT2AALDH1A1HSD17B10
SCHEMBL11990862 0.74 ALDH1A1 (0.70) RAB9AMEN1KMT2AALDH1A1NPC1
SCHEMBL12341700 0.74 ESR1 (0.63) RAB9AMEN1KMT2AALDH1A1NPC1
SCHEMBL16965593 0.72 NPSR1 (0.48) MEN1KMT2AALDH1A1TSHRL3MBTL1
SCHEMBL20735076 0.71 RAB9A (0.52) RAB9AMEN1KMT2AALDH1A1HSD17B10
SCHEMBL20735114 0.71 RAB9A (0.52) RAB9AMEN1KMT2AALDH1A1HSD17B10
SCHEMBL13400255 0.70 MEN1 (0.71) RAB9AMEN1KMT2AALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900239-B1 DIHYDRO-6-AZAPHENALENE DERIVATIVES FOR THE TREATMENT OF CNS, OCULAR DISEASES AND RELATED DISORDERS WARNER BABCOCK INST FOR GREEN CHEMISTRY LLC (US) 2019-03-20 EP disclosed