SCHEMBL2083165

SCHEMBL2083165

O=Cc1cc2ccc(Br)cc2s1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 8/20 0.58
ERN1 O75460 2/20 0.42
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
CHRNA7 P36544 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
DYRK1A Q13627 1/20 0.34
DHPS P49366 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30197462 1.00 CYP2A6 (0.58) CYP2A6ERN1NPC1RAB9AALDH1A1
SCHEMBL2019385 0.85 CYP2A6 (0.62) CYP2A6ERN1RAB9AALDH1A1DYRK1A
SCHEMBL23775695 0.78 CYP2A6 (0.60) CYP2A6RAB9AALDH1A1
SCHEMBL4385517 0.77 CYP2A6 (0.58) CYP2A6ERN1NPC1RAB9AALDH1A1
SCHEMBL21234909 0.77 CYP2A6 (0.58) CYP2A6MAPTHTT
SCHEMBL6963606 0.77 CYP2A6 (0.58) CYP2A6NPC1RAB9AALDH1A1MAPT
SCHEMBL20391352 0.77 CYP2A6 (0.58) CYP2A6ALDH1A1
SCHEMBL28086785 0.77 CYP2A6 (0.73) CYP2A6NPC1RAB9AALDH1A1MAPT
SCHEMBL12683402 0.77 CYP2A6 (0.61) CYP2A6
SCHEMBL7972992 0.77 RAB9A (0.38) CYP2A6ERN1NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117305308-A High-stability nucleic acid aptamer molecule, and compound and application thereof 华东理工大学 2023-12-29 CN disclosed
EP-3647311-B1 RHO-ASSOCIATED PROTEIN KINASE INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD AND USE THEREOF BEIJING TIDE PHARMACEUTICAL CO LTD (CN) 2023-11-01 EP disclosed
CN-115974762-B Diamine monomer with bulky alkynyl side group, polybenzoxazole precursor, photosensitive resin composition and application thereof 波米科技有限公司 2023-09-19 CN disclosed
CN-115626890-B Diamine monomer with bulky alkynyl side group, and preparation method and application thereof 波米科技有限公司 2023-05-16 CN disclosed
CN-115974762-A Diamine monomer with bulky alkynyl side group, polybenzoxazole precursor, photosensitive resin composition and application thereof 波米科技有限公司 2023-04-18 CN disclosed
CN-115704025-A Novel nucleic acid molecule detection and quantification technology 华东理工大学 2023-02-17 CN disclosed
CN-115626890-A Diamine monomer with bulky alkynyl side group and preparation method and application thereof 波米科技有限公司 2023-01-20 CN disclosed
EP-3421465-B1 RHO-ASSOCIATED PROTEIN KINASE INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AS WELL AS PREPARATION METHOD AND USE THEREOF BEIJING TIDE PHARMACEUTICAL CO LTD (CN) 2022-10-26 EP disclosed
CN-111592472-B Fluorescent dye and preparation method and application thereof 纳莹(上海)生物科技有限公司 2022-10-21 CN disclosed
EP-3421464-B1 RHO-ASSOCIATED PROTEIN KINASE INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AS WELL AS PREPARATION METHOD AND USE THEREOF BEIJING TIDE PHARMACEUTICAL CO LTD (CN) 2021-11-24 EP disclosed
US-7863302-B2 Compounds and methods for modulating FX-receptors ELI LILLY AND COMPANY (US) 2011-01-04 US disclosed
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION 2010-09-02 US disclosed
US-20080306125-A1 Compounds and Methods for Modulating Fx-Receptors JPMORGAN CHASE BANK, N.A., AS SUCCESSOR COLLATERAL AGENT 2008-12-11 US disclosed
EP-1984360-A2 COMPOUNDS AND METHODS FOR MODULATING FX-RECEPTORS Eli Lilly & Company (US) 2008-10-29 EP disclosed
US-7339065-B2 Design and synthesis of optimized ligands for PPAR BETHESDA PHARMACEUTICALS, INC. (US) 2008-03-04 US disclosed
US-7339065-B2 Design and synthesis of optimized ligands for PPAR BETHESDA PHARMACEUTICALS, INC. (US) 2008-03-04 US disclosed
WO-2007092751-A2 COMPOUNDS AND METHODS FOR MODULATING FX-RECEPTORS ELI LILLY AND COMPANY (US) 2007-08-16 WO disclosed
US-20070099969-A1 Design and synthesis of optimized ligands for ppar THE UNIVERSITY OF MISSISSIPPI 2007-05-03 US disclosed
US-20070099969-A1 Design and synthesis of optimized ligands for ppar THE UNIVERSITY OF MISSISSIPPI 2007-05-03 US disclosed
WO-2001090105-A1 ISOTHIAZOLES AS PESTICIDES SYNGENTA LIMITED (GB) 2001-11-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080306125-A1 Compounds and Methods for Modulating Fx-Receptors F2R, TBXA2R, PTAFR CYP2A6 731/4885ERN1 3507/4885NPC1 426/4885
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS OPRL1, OPRM1, OPRK1 CYP2A6 1871/4885ERN1 2555/4885NPC1 2935/4885
US-20070099969-A1 Design and synthesis of optimized ligands for ppar PPARD, PPARA, PPARG CYP2A6 133/4885ERN1 4155/4885NPC1 2436/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.