SCHEMBL20839740

SCHEMBL20839740

CCOC(=O)CCc1cccc(NC(=O)c2ccccc2NC(=O)C#Cc2ccccc2)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 7/20 0.50
PPARG P37231 5/20 0.50
PPARA Q07869 5/20 0.50
PPARD Q03181 6/20 0.48
RXFP1 Q9HBX9 3/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
GFER P55789 1/20 0.43
BRD4 O60885 1/20 0.42
MAPT P10636 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
F2R P25116 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20839715 0.87 NR1H4 (0.61) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL20839943 0.78 FADS1 (0.52) NR1H4PPARGPPARAABCG2SIRT2
SCHEMBL7457415 0.76 SIRT2 (0.53) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL20839724 0.75 CYP3A4 (0.52) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL20839629 0.75 NR1H4 (0.56) NR1H4PPARGPPARAPPARDABCG2
SCHEMBL20839494 0.75 NR1H4 (0.45) NR1H4PPARGPPARAPPARDRXFP1
SCHEMBL20839484 0.75 ABCG2 (0.68) ABCG2MEN1KMT2AMAPTALDH1A1
SCHEMBL20839668 0.74 NR1H4 (0.56) NR1H4PPARGPPARAPPARDRXFP1
SCHEMBL15591247 0.72 PTGER4 (0.49) NR1H4MEN1KMT2ABRD4MAPT
SCHEMBL20852275 0.72 NR1H4 (0.71) NR1H4PPARGPPARAPPARDRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed