SCHEMBL20852275

SCHEMBL20852275

CC(=O)Nc1ccccc1C(=O)Nc1cccc(CCC(=O)O)c1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 10/20 0.71
PPARG P37231 7/20 0.71
PPARA Q07869 7/20 0.71
PPARD Q03181 9/20 0.68
RXFP1 Q9HBX9 1/20 0.58
SIRT1 Q96EB6 1/20 0.58
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
ABCG2 Q9UNQ0 1/20 0.55
ITGB3 P05106 1/20 0.54
ITGA2B P08514 1/20 0.54
ALDH1A1 P00352 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
HSPH1 Q92598 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10752853 0.84 MEN1 (0.61) NR1H4PPARGPPARASIRT1MEN1
SCHEMBL20852079 0.84 NR1H4 (0.81) NR1H4PPARGPPARAPPARDRXFP1
SCHEMBL5718041 0.82 ALOX15 (0.72) NR1H4PPARGPPARAPPARDSIRT1
SCHEMBL20839783 0.82 NR1H4 (0.80) NR1H4PPARGPPARAPPARDRXFP1
SCHEMBL20839715 0.82 NR1H4 (0.61) NR1H4PPARGPPARAPPARDSIRT1
SCHEMBL20839480 0.81 ITGB3 (0.60) NR1H4PPARGPPARAPPARDSIRT1
SCHEMBL27134473 0.80 KMT2A (0.77) RXFP1MEN1KMT2AALDH1A1
SCHEMBL7450542 0.79 ITGB3 (0.72) NR1H4PPARGPPARAPPARDSIRT1
SCHEMBL16088635 0.79 ALDH1A1 (0.60) NR1H4PPARGPPARAPPARDMEN1
SCHEMBL20839733 0.78 NR1H4 (0.72) NR1H4PPARGPPARAPPARDRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed