SCHEMBL20839965

SCHEMBL20839965

O=C(O)CCc1cccc(NC(=O)c2ccccc2NC(=O)C2=C(Cl)c3ccccc3OC2)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 11/20 0.56
PPARD Q03181 10/20 0.56
PPARG P37231 8/20 0.56
PPARA Q07869 8/20 0.56
HSPH1 Q92598 1/20 0.51
SIRT1 Q96EB6 1/20 0.45
TP53 P04637 1/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
CYP3A4 P08684 1/20 0.44
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
GRM5 P41594 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20839494 0.88 NR1H4 (0.45) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839742 0.81 NR1H4 (0.57) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839654 0.79 MEN1 (0.62) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839983 0.78 NR1H4 (0.56) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839719 0.77 NR1H4 (0.54) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839968 0.76 NR1H4 (0.56) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20852275 0.76 NR1H4 (0.71) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20852079 0.74 NR1H4 (0.81) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839783 0.73 NR1H4 (0.80) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839715 0.73 NR1H4 (0.61) NR1H4PPARDPPARGPPARAHSPH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed