SCHEMBL20867962

SCHEMBL20867962

CCOC(=O)CN(C)CC1COC(C)(C)N1C(=O)OC(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SPHK1 Q9NYA1 1/20 0.43
BRD4 O60885 1/20 0.34
HSD11B2 P80365 1/20 0.33
GLA P06280 1/20 0.31
HCRTR2 O43614 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21455299 1.00 SPHK1 (0.43) SPHK1BRD4HSD11B2GLAHCRTR2
SCHEMBL21455156 1.00 SPHK1 (0.43) SPHK1BRD4HSD11B2GLAHCRTR2
SCHEMBL8445237 0.81 SPHK1 (0.46) SPHK1BRD4HSD11B2GLAHCRTR2
SCHEMBL14357932 0.81 SPHK1 (0.46) SPHK1BRD4HSD11B2GLAHCRTR2
SCHEMBL7500054 0.81 SPHK1 (0.38) SPHK1BRD4HSD11B2
SCHEMBL7500049 0.81 SPHK1 (0.38) SPHK1BRD4HSD11B2
SCHEMBL6719410 0.80 SPHK1 (0.37) SPHK1BRD4L3MBTL1MEN1KMT2A
SCHEMBL7499191 0.80 SPHK1 (0.37) SPHK1BRD4L3MBTL1MEN1KMT2A
SCHEMBL7499187 0.80 SPHK1 (0.37) SPHK1BRD4L3MBTL1MEN1KMT2A
SCHEMBL3465657 0.80 SPHK1 (0.44) SPHK1BRD4HSD11B2GLAHCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10934311-B2 Heterocyclic compound used as FGFR inhibitor HANGZHOU INNOGATE PHARMA CO., LTD. (CN) 2021-03-02 US disclosed
US-20190100531-A1 HETEROCYCLIC COMPOUND USED AS FGFR INHIBITOR HANGZHOU INNOGATE PHARMA CO., LTD. (CN) 2019-04-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190100531-A1 HETEROCYCLIC COMPOUND USED AS FGFR INHIBITOR FGFR1, FGFR3, FGFR2 SPHK1 2674/4885BRD4 138/4885HSD11B2 192/4885
US-10934311-B2 Heterocyclic compound used as FGFR inhibitor FGFR1, FGFR3, FGFR2 SPHK1 2674/4885BRD4 138/4885HSD11B2 192/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.