SCHEMBL20870488

SCHEMBL20870488

COC(=O)c1cc(N=O)ccc1OCC1CCOCC1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RORC P51449 7/20 0.44
SCN9A Q15858 1/20 0.42
XDH P47989 1/20 0.41
IRAK4 Q9NWZ3 2/20 0.40
BRD4 O60885 1/20 0.40
GRM4 Q14833 3/20 0.38
P2RX4 Q99571 3/20 0.38
PTGER1 P34995 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20870201 0.84 RORC (0.46) RORCSCN9AXDHIRAK4BRD4
SCHEMBL20870215 0.83 RORC (0.45) RORCSCN9AXDHIRAK4BRD4
SCHEMBL22297975 0.83 RORC (0.54) RORCSCN9ABRD4
SCHEMBL20870409 0.83 RORC (0.49) RORCSCN9AXDHBRD4
SCHEMBL28715124 0.82 BRD4 (0.45) RORCSCN9AXDHBRD4P2RX4
SCHEMBL20870218 0.81 RORC (0.46) RORCSCN9AXDHIRAK4BRD4
SCHEMBL22262327 0.80 ALDH1A1 (0.52) SCN9ABRD4
SCHEMBL20529251 0.80 RORC (0.51) RORCSCN9AP2RX4
SCHEMBL20870210 0.80 RORC (0.51) RORCSCN9AP2RX4
SCHEMBL28715152 0.80 BRD4 (0.43) RORCSCN9AXDHBRD4OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019063015-A1 SULFONYL-SUBSTITUTED BICYCLIC COMPOUND WHICH ACTS AS RORγ INHIBITOR 正大天晴药业集团股份有限公司 2019-04-04 WO disclosed