SCHEMBL20908009

SCHEMBL20908009

CC(C)OC(=O)[C@@](N)(CC(C)(C)C)c1ccc(Br)cc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 3/20 0.36
DGAT1 O75907 1/20 0.35
APLNR P35414 4/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
MAPT P10636 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
FPR2 P25090 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MCL1 Q07820 1/20 0.32
MAPK1 P28482 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28401181 1.00 AAK1 (0.36) AAK1DGAT1APLNRNPC1RAB9A
SCHEMBL21150265 0.84 KIF11 (0.43) NPC1RAB9ASMN1; SMN2L3MBTL1
SCHEMBL20907524 0.84 KIF11 (0.43) NPC1RAB9ASMN1; SMN2L3MBTL1
Hydrochloric Acid SCHEMBL28401748 0.83 KIF11 (0.42) NPC1RAB9ASMN1; SMN2L3MBTL1
SCHEMBL28407437 0.83 MAP2K1 (0.32)
SCHEMBL20907832 0.83 MAP2K1 (0.32)
Hydrochloric Acid SCHEMBL28401746 0.83 KIF11 (0.42) NPC1RAB9ASMN1; SMN2L3MBTL1
SCHEMBL21112403 0.82 DGAT1 (0.41) AAK1DGAT1NPC1RAB9ASMN1; SMN2
SCHEMBL21112405 0.82 DGAT1 (0.41) AAK1DGAT1NPC1RAB9ASMN1; SMN2
SCHEMBL30557344 0.82 DGAT1 (0.41) AAK1DGAT1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11352329-B2 HIV protease inhibitors GILEAD SCIENCES, INC. (US) 2022-06-07 US disclosed
CN-111212832-A 1-benzyl-2-imino-4-phenyl-5-oxoimidazolidine derivatives as HIV protease inhibitors 吉利德科学公司 2020-05-29 CN disclosed
WO-2019075291-A1 1-BENZYL-2-IMINO-4-PHENYL-5-OXOIMIDAZOLIDINE DERIVATIVES AS HIV PROTEASE INHIBITORS GILEAD SCIENCES, INC. (US) 2019-04-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11352329-B2 HIV protease inhibitors PRSS1, SERPINB1, FURIN AAK1 1993/4885DGAT1 3349/4885APLNR 3099/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.