SCHEMBL20910192

SCHEMBL20910192

Cc1ccc2c(c1)CN(CC(=O)N(C)C)CC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
ALDH1A1 P00352 4/20 0.47
NPSR1 Q6W5P4 1/20 0.47
DRD2 P14416 4/20 0.44
KDM4E B2RXH2 5/20 0.44
TSHR P16473 2/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
GAA P10253 1/20 0.43
RAB9A P51151 1/20 0.43
GFER P55789 1/20 0.43
DRD3 P35462 2/20 0.41
SIGMAR1 Q99720 1/20 0.41
NOTUM Q6P988 1/20 0.41
AKR1C3 P42330 1/20 0.41
MAPT P10636 2/20 0.40
POLB P06746 1/20 0.40
XIAP P98170 1/20 0.40
BIRC2 Q13490 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13345546 0.84 MEN1 (0.52) MEN1KMT2AALDH1A1NPSR1DRD2
SCHEMBL24192767 0.83 KMT2A (0.51) MEN1KMT2AALDH1A1NPSR1DRD2
SCHEMBL20889996 0.83 XIAP (0.43) MEN1KMT2ADRD2RAB9AGFER
SCHEMBL24478514 0.83 HTR5A (0.46) MEN1KMT2AALDH1A1NPSR1DRD2
SCHEMBL22549193 0.80 CHRM2 (0.53) MEN1KMT2AALDH1A1NPSR1DRD2
SCHEMBL22543662 0.79 DRD2 (0.39) MEN1KMT2ADRD2RAB9AGFER
SCHEMBL24478527 0.77 KIF11 (0.34) MEN1KMT2ADRD2KDM4EXIAP
SCHEMBL24478250 0.77 DRD2 (0.45) MEN1KMT2AALDH1A1DRD2KDM4E
SCHEMBL15756197 0.76 KMT2A (0.55) MEN1KMT2AALDH1A1DRD2KDM4E
SCHEMBL521473 0.76 DRD2 (0.57) ALDH1A1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020210380-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF NUVATION BIO INC. (US) 2020-10-15 WO disclosed
WO-2019074979-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF GIRAFPHARMA, LLC (US) 2019-04-18 WO disclosed