SCHEMBL20919681

SCHEMBL20919681

COC(=O)c1ccc(F)c(OC2CCCC2)c1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 14/20 0.55
PDE4B Q07343 11/20 0.55
PDE4A P27815 10/20 0.55
PDE4C Q08493 10/20 0.55
EPHX2 P34913 1/20 0.54
PDE5A O76074 1/20 0.50
MAPK14 Q16539 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15904302 0.89 PDE4D (0.55) PDE4DPDE4BPDE4APDE4CPDE5A
SCHEMBL1409231 0.85 ALOX15 (0.53) PDE4DPDE4BPDE4APDE4CEPHX2
SCHEMBL5309884 0.84 PDE4D (0.67) PDE4DPDE4BPDE4APDE4CPDE5A
SCHEMBL7364684 0.84 PDE4D (0.60) PDE4DPDE4BPDE4APDE4CPDE5A
SCHEMBL7355374 0.84 CA12 (0.54) PDE4DPDE4BPDE4APDE4CPDE5A
SCHEMBL1409590 0.84 PDE4D (0.53) PDE4DPDE4BPDE4APDE4CEPHX2
SCHEMBL28650035 0.83 PDE4B (0.50) PDE4DPDE4BPDE4APDE4CEPHX2
SCHEMBL7360312 0.82 PDE4D (0.68) PDE4DPDE4BPDE4APDE4CPDE5A
SCHEMBL27372082 0.82 PDE4D (0.52) PDE4DPDE4BPDE4APDE4CEPHX2
SCHEMBL7358414 0.81 PDE4D (0.55) PDE4DPDE4BPDE4APDE4CEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11572347-B2 Orally available sEH/PDE4 dual inhibitors THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-02-07 US disclosed
US-11572347-B2 Orally available sEH/PDE4 dual inhibitors THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-02-07 US disclosed
US-20210395202-A1 ORALLY AVAILABLE SEH/PDE4 DUAL INHIBITORS GOETHE-UNIVERSITY FRANKFURT (DE) 2021-12-23 US disclosed
US-20210395202-A1 ORALLY AVAILABLE SEH/PDE4 DUAL INHIBITORS GOETHE-UNIVERSITY FRANKFURT (DE) 2021-12-23 US disclosed
WO-2019079609-A1 ORALLY AVAILABLE SEH/PDE4 DUAL INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-04-25 WO disclosed
WO-2019079609-A1 ORALLY AVAILABLE SEH/PDE4 DUAL INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-04-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11572347-B2 Orally available sEH/PDE4 dual inhibitors EPHX1, PDE4A, EPHX2 PDE4D 14/4885PDE4B 5/4885PDE4A 2/4885
US-20210395202-A1 ORALLY AVAILABLE SEH/PDE4 DUAL INHIBITORS EPHX1, PDE4A, EPHX2 PDE4D 14/4885PDE4B 5/4885PDE4A 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.