SCHEMBL20969307

SCHEMBL20969307

N[C@@H](c1c(F)cccc1F)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.36
CES1 P23141 2/20 0.36
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
MC4R P32245 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20531764 1.00 CES2 (0.36) CES2CES1HTR2AHTR2CMC4R
SCHEMBL21884017 0.86 ACHE (0.41) CES2CES1HTR2AHTR2C
SCHEMBL19768998 0.82 HTR2C (0.36) HTR2AHTR2C
SCHEMBL21884016 0.81 HTR2A (0.30) HTR2AHTR2C
SCHEMBL19880513 0.81 GABRA1 (0.39) CES2CES1HTR2AHTR2CMC4R
SCHEMBL19880514 0.77 TSHR (0.40) HTR2AHTR2CMC4R
SCHEMBL18306095 0.74 CYP1A2 (0.38)
SCHEMBL20238028 0.74 IDO1 (0.41) CES2CES1
SCHEMBL20238027 0.74 IDO1 (0.41) CES2CES1
SCHEMBL29669053 0.74 IDO1 (0.41) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3481823-A1 7-SUBSTITUTED 1-PYRIDYL-NAPHTHYRIDINE-3-CARBOXYLIC ACID AMIDES AND USE THEREOF Bayer Pharma Aktiengesellschaft (DE) 2019-05-15 EP disclosed