SCHEMBL20977928

SCHEMBL20977928

Bn1cncc1C(=O)N(C)OC

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.35
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
MLYCD O95822 1/20 0.33
ICAM1 P05362 1/20 0.31
SELE P16581 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
CLK1 P49759 1/20 0.31
DYRK1A Q13627 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3450620 0.81 CYP11B1 (0.36) MAPK1CYP11B1CYP11B2MLYCDICAM1
SCHEMBL18137641 0.71 TBXAS1 (0.44) CYP11B2
SCHEMBL24966165 0.70 MAPK1 (0.70) MAPK1CYP11B1CYP11B2GPBAR1
SCHEMBL23234282 0.70 MAPK1 (0.70) MAPK1CYP11B1CYP11B2GPBAR1
SCHEMBL18137637 0.69 SLC6A3 (0.36) MAPK1CYP11B1CYP11B2MLYCD
SCHEMBL18137612 0.69 IDO1 (0.40) ICAM1SELE
SCHEMBL16462029 0.68 HSD11B1 (0.35) MLYCDICAM1SELETRPM8CLK1
SCHEMBL2507311 0.67 HCAR2 (0.46) MLYCDICAM1SELETRPM8CLK1
SCHEMBL20305483 0.65 ESR1 (0.44) MLYCDICAM1SELETRPM8CLK1
SCHEMBL14937988 0.64 HTT (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2814814-B1 IMIDAZOLYLKETONE DERIVATIVES ASD ALDOSTERONE SYNTHASE INHIBITORS HOFFMANN LA ROCHE (CH) 2019-05-08 EP disclosed