SCHEMBL20998615

SCHEMBL20998615

CC(=O)CCCCNC(N)=S

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PAOX Q6QHF9 8/20 0.50
ADRA1A P35348 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MAPK1 P28482 1/20 0.43
HIF1A Q16665 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TAS2R38 P59533 1/20 0.38
PRMT1 Q99873 1/20 0.38
ALDH1A1 P00352 1/20 0.36
EPHX2 P34913 1/20 0.36
ACHE P22303 1/20 0.35
CASP2 P42575 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL377237 0.83 EPHX2 (0.49) PAOXADRA1AKDM4EMAPK1HIF1A
SCHEMBL12962267 0.83 PAOX (0.53) PAOXADRA1AKDM4EMAPK1HIF1A
SCHEMBL26748554 0.81 PAOX (0.57) PAOXADRA1AKDM4EMAPK1HIF1A
SCHEMBL28444812 0.81 PAOX (0.57) PAOXADRA1AKDM4EMAPK1HIF1A
SCHEMBL10287837 0.79 PAOX (0.50) PAOXADRA1AKDM4EMAPK1HIF1A
SCHEMBL18256338 0.79 FAAH (0.55) MEN1KMT2AEPHX2CASP2
SCHEMBL381238 0.79 EPHX2 (0.50) ALDH1A1EPHX2
SCHEMBL13902111 0.78 KDM4E (0.71) PAOXADRA1AKDM4EMAPK1HIF1A
SCHEMBL23571063 0.78 PAOX (0.53) PAOXADRA1AKDM4EMAPK1HIF1A
SCHEMBL12119633 0.78 PAOX (0.53) PAOXADRA1AKDM4EMAPK1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060550-B1 HETEROARYL COMPOUNDS AS BTK INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2019-05-15 EP disclosed
CN-103025710-A Process for the synthesis of isothiocyanates and derivatives thereof and uses of same AURIGA INTERNAT 2013-04-03 CN disclosed