SCHEMBL377237

SCHEMBL377237

CC(=O)CCCCNC(=S)NCCCCC(C)=O

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 7/20 0.49
PAOX Q6QHF9 6/20 0.48
ADRA1A P35348 1/20 0.47
KDM4E B2RXH2 1/20 0.46
MAPK1 P28482 1/20 0.46
HIF1A Q16665 1/20 0.46
PRMT1 Q99873 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SIRT5 Q9NXA8 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26748552 0.88 PAOX (0.47) EPHX2PAOXADRA1AKDM4EMAPK1
SCHEMBL459515 0.86 EPHX2 (0.40) EPHX2PAOXADRA1AKDM4EMAPK1
SCHEMBL28801749 0.86 EPHX2 (0.43) EPHX2PAOXADRA1AKDM4EMAPK1
SCHEMBL373838 0.84 EPHX2 (0.39) EPHX2PAOXADRA1AKDM4EMAPK1
SCHEMBL20998615 0.83 PAOX (0.50) EPHX2PAOXADRA1AKDM4EMAPK1
SCHEMBL13902111 0.81 KDM4E (0.71) PAOXADRA1AKDM4EMAPK1HIF1A
Thiourea SCHEMBL14990305 0.80 PAOX (0.38) EPHX2PAOXADRA1AKDM4EMAPK1
SCHEMBL14990106 0.79 PAOX (0.43) EPHX2PAOXADRA1AKDM4EMAPK1
SCHEMBL24572062 0.79 KDM4E (0.76) PAOXADRA1AKDM4EMAPK1HIF1A
SCHEMBL6427110 0.79 ADRA1A (0.54) PAOXADRA1AKDM4EMAPK1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214188-A1 COMPOSITIONS FOR STABILIZING AN ISOTHIOCYANATE VIO CHEMICALS AG (CH) 2021-10-28 WO disclosed
US-20130142739-A1 PROCESS FOR THE SYNTHESIS OF ISOTHIOCYANATES AND DERIVATIVES THEREOF AND USES OF SAME AURIGA INTERNATIONAL (BE) 2013-06-06 US disclosed
US-20130142739-A1 PROCESS FOR THE SYNTHESIS OF ISOTHIOCYANATES AND DERIVATIVES THEREOF AND USES OF SAME AURIGA INTERNATIONAL (BE) 2013-06-06 US disclosed
US-20130142739-A1 PROCESS FOR THE SYNTHESIS OF ISOTHIOCYANATES AND DERIVATIVES THEREOF AND USES OF SAME AURIGA INTERNATIONAL (BE) 2013-06-06 US disclosed
WO-2012010644-A1 PROCESS FOR THE SYNTHESIS OF ISOTHIOCYANATES AND DERIVATIVES THEREOF AND USES OF SAME AURIGA INTERNATIONAL (BE) 2012-01-26 WO disclosed
EP-2409693-A2 Isothiocyanates and derivatives for use in the treatment and / or prevention of polymorphous light eruptions Auriga International (BE) 2012-01-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130142739-A1 PROCESS FOR THE SYNTHESIS OF ISOTHIOCYANATES AND DERIVATIVES THEREOF AND USES OF SAME TST, CBS, SRM EPHX2 2218/4885PAOX 3642/4885ADRA1A 3447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.